Identification of sulfonamide based butyrylcholinesterase inhibitors through scaffold hopping approach
Ankit Ganeshpurkar, Ravi Singh, Devendra Kumar, Pravin Gore, Shalini Shivhare, Divya Sardana, Rayala Swetha, Ashok Kumar, Sushil Kumar Singh
Topics & Concepts
ButyrylcholinesteraseChemistryAcetylcholinesteraseAcetamidePharmacophoreBenzamideStereochemistryEnzymeAchéCholinesteraseDocking (animal)BiochemistryPharmacologyOrganic chemistryBiologyNursingMedicineCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsEnzyme function and inhibition