Schiff bases of 4-Phenyl-2-Aminothiazoles as hits to new antischistosomals: Synthesis, in vitro, in vivo and in silico studies
Carina R. Amorim, Thais Fernanda Amorim Pavani, Andrey F.S. Lopes, Marcelo Dutra Duque, Ana C. Mengarda, Marcos P. Silva, Josué de Moraes, Daniela Rando
Topics & Concepts
In vivoBioavailabilityChemistryIn silicoPharmacologyIn vitroSchistosoma mansoniDrugBiochemistryThiazolePharmacokineticsProtein tyrosine phosphataseIC50BiologyKinaseStereochemistrySchistosomiasisImmunologyBiotechnologyHelminthsGeneParasites and Host InteractionsResearch on Leishmaniasis StudiesHelminth infection and control