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Myricetin reduces cytotoxicity by suppressing hepcidin expression in MES23.5 cells

Han Deng, Shang Liu, Dong Pan, Yi Jia, Zegang Ma

2020Neural Regeneration Research22 citationsDOIOpen Access PDF

Abstract

M myricetin for 1 hour, followed by co-treatment with 400 nM rotenone for 24 hours to establish an in vitro cell model of Parkinson's disease. Our results revealed that myricetin alleviated rotenone-induced decreases in cell viability, suppressed the production of intracellular reactive oxygen species, and restored mitochondrial transmembrane potential. In addition, myricetin significantly suppressed rotenone-induced hepcidin gene transcription and partly relieved rotenone-induced inhibition of ferroportin 1 mRNA and protein levels. Furthermore, myricetin inhibited rotenone-induced phosphorylation of STAT3 and SMAD1 in MES23.5 cells. These findings suggest that myricetin protected rotenone-treated MES23.5 cells by potently inhibiting hepcidin expression to prevent iron accumulation, and this effect was mediated by alteration of STAT3 and SMAD1 signaling pathways.

Topics & Concepts

RotenoneMyricetinNeuroprotectionViability assayHepcidinSubstantia nigraReactive oxygen speciesChemistryPharmacologyOxidative stressCell biologyIntracellularBiochemistryBiologyApoptosisMitochondrionAntioxidantInflammationDopaminergicEndocrinologyImmunologyDopamineFlavonoidKaempferolIron Metabolism and DisordersTrace Elements in HealthRNA regulation and disease