Structure-guided identification of novel dual-targeting estrogen receptor α degraders with aromatase inhibitory activity for the treatment of endocrine-resistant breast cancer
Lilan Xin, Jian Min, Hebing Hu, Yuanyuan Li, Chuanqian Du, Baohua Xie, Yan Cheng, Xiaofei Deng, Xiangping Deng, Kang Shen, Jian Huang, Chun‐Chi Chen, Rey‐Ting Guo, Chune Dong, Hai‐Bing Zhou
Topics & Concepts
AromataseEstrogen receptorChemistryCancer researchEstrogen receptor alphaEstrogenSelective estrogen receptor modulatorBreast cancerPharmacologyCancerInternal medicineEndocrinologyBiologyMedicineEstrogen and related hormone effectsHistone Deacetylase Inhibitors ResearchProtein Degradation and Inhibitors