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Property activity refinement of 2-anilino 4-amino substituted quinazolines as antimalarials with fast acting asexual parasite activity

Trent D. Ashton, Anna Ngo, Paola Favuzza, Hayley E. Bullen, Maria R. Gancheva, Ornella Romeo, Molly Parkyn Schneider, Nghi Nguyen, Ryan Steel, Sandra Duffy, Kym N. Lowes, Hélène Jousset Sabroux, Vicky M. Avery, Justin A. Boddey, Danny W. Wilson, Alan F. Cowman, Paul R. Gilson, Brad E. Sleebs

2021Bioorganic Chemistry20 citationsDOIOpen Access PDF

Topics & Concepts

QuinazolinePlasmodium falciparumMalariaCytotoxicityChemistryGametocytePlasmodium bergheiIn vitroIndolineBiochemistryBiologyPharmacologyCombinatorial chemistryStereochemistryImmunologyMalaria Research and ControlQuinazolinone synthesis and applicationsMosquito-borne diseases and control
Property activity refinement of 2-anilino 4-amino substituted quinazolines as antimalarials with fast acting asexual parasite activity | Litcius