Property activity refinement of 2-anilino 4-amino substituted quinazolines as antimalarials with fast acting asexual parasite activity
Trent D. Ashton, Anna Ngo, Paola Favuzza, Hayley E. Bullen, Maria R. Gancheva, Ornella Romeo, Molly Parkyn Schneider, Nghi Nguyen, Ryan Steel, Sandra Duffy, Kym N. Lowes, Hélène Jousset Sabroux, Vicky M. Avery, Justin A. Boddey, Danny W. Wilson, Alan F. Cowman, Paul R. Gilson, Brad E. Sleebs
Topics & Concepts
QuinazolinePlasmodium falciparumMalariaCytotoxicityChemistryGametocytePlasmodium bergheiIn vitroIndolineBiochemistryBiologyPharmacologyCombinatorial chemistryStereochemistryImmunologyMalaria Research and ControlQuinazolinone synthesis and applicationsMosquito-borne diseases and control