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Allosteric Activation of PI3Kα Results in Dynamic Access to Catalytically Competent Conformations

Mayukh Chakrabarti, Sandra B. Gabelli, L. Mario Amzel

2020Structure20 citationsDOIOpen Access PDF

Topics & Concepts

Allosteric regulationChemistryComputational biologyBiochemistryEnzymeBiophysicsBiologyPI3K/AKT/mTOR signaling in cancerChronic Lymphocytic Leukemia ResearchBiochemical and Molecular Research
Allosteric Activation of PI3Kα Results in Dynamic Access to Catalytically Competent Conformations | Litcius