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Reprofiling of approved drugs against SARS-CoV-2 main protease: an in-silico study

Prateek Kumar, Taniya Bhardwaj, Ankur Kumar, Bhuvaneshwari R. Gehi, Shivani Krishna Kapuganti, Neha Garg, Gopal Nath, Rajanish Giri

2020Journal of Biomolecular Structure and Dynamics26 citationsDOIOpen Access PDF

Abstract

. We believe that the high-affinity binding of these compounds will help in designing novel strategies for structure-based drug discovery against SARS-CoV-2.Communicated by Ramaswamy H. Sarma.

Topics & Concepts

In silicoProteaseRepurposingDocking (animal)Drug repositioningVirtual screeningPharmacologyDrug discoveryDrugEndoribonucleaseChemistryVirologyComputational biologyBiologyBiochemistryMedicineEnzymeRNAGeneEcologyRNase PNursingComputational Drug Discovery MethodsSARS-CoV-2 and COVID-19 ResearchProtein Structure and Dynamics
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