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Organophotoredox-Catalyzed Three-Component Coupling of Heteroatom Nucleophiles, Alkenes, and Aliphatic Redox Active Esters

Shotaro Shibutani, Kazunori Nagao, Hirohisa Ohmiya

2021Organic Letters80 citationsDOI

Abstract

This manuscript describes a visible-light-mediated organophotoredox catalytic process for vicinal difunctionalization of alkenes using heteroatom nucleophiles and aliphatic redox active esters. A wide range of heteroatom nucleophiles including alcohols, water, carboxylic acids, amides, and halogens can be used for this reaction. This radical relay type reaction allows forging of C(sp3)–C(sp3) with a carbon-centered radical and C(sp3)–heteroatom bonds with a benzyl cation on the vinylarenes with complete regioselectivity in a single step.

Topics & Concepts

ChemistryNucleophileHeteroatomRegioselectivityCatalysisVicinalRedoxHalogenCoupling reactionReactivity (psychology)Organic chemistryCombinatorial chemistryMedicinal chemistryRing (chemistry)AlkylMedicinePathologyAlternative medicineRadical Photochemical ReactionsSulfur-Based Synthesis TechniquesCatalytic C–H Functionalization Methods
Organophotoredox-Catalyzed Three-Component Coupling of Heteroatom Nucleophiles, Alkenes, and Aliphatic Redox Active Esters | Litcius