Litcius/Paper detail

Imidazo[1,2-a]quinazolines as novel, potent EGFR-TK inhibitors: Design, synthesis, bioactivity evaluation, and in silico studies

Zaman Hasanvand, Tayebeh Oghabi Bakhshaiesh, Fariba Peytam, Loghman Firoozpour, Elaheh Hosseinzadeh, Rasoul Motahari, Setareh Moghimi, Elaheh Nazeri, Mahsa Toolabi, Farhad Momeni, Hamid Reza Bijanzadeh, Ali Khalaj, Blandine Baratte, Béatrice Josselin, Thomas Robert, Stéphane Bach, Rezvan Esmaeili, Alireza Foroumadi

2023Bioorganic Chemistry17 citationsDOI

Topics & Concepts

ChemistryIn silicoPharmacologyEGFR inhibitorsComputational biologyCombinatorial chemistryBiochemistryEpidermal growth factor receptorReceptorGeneBiologyMedicineQuinazolinone synthesis and applicationsLung Cancer Treatments and MutationsSynthesis and Biological Evaluation