Effect of the dichloro-substitution on antiproliferative activity of phthalimide-thiazole derivatives. Rational design, synthesis, elastase, caspase 3/7, and EGFR tyrosine kinase activity and molecular modeling study
Beata Donarska, Marta Świtalska, Wojciech Płaziński, Joanna Wietrzyk, Krzysztof Z. Łączkowski
Topics & Concepts
ChemistryTyrosine kinaseThiazoleElastasePhthalimideSubstitution (logic)KinaseBiochemistryStereochemistryPharmacologyCombinatorial chemistryEnzymeSignal transductionComputer scienceMedicineProgramming languageSynthesis and biological activityCytokine Signaling Pathways and InteractionsHER2/EGFR in Cancer Research