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Design, green synthesis, molecular docking and anticancer evaluations of diazepam bearing sulfonamide moieties as VEGFR-2 inhibitors

Nashwa M. Saleh, Mohamed S.A. El-Gaby, Khaled El‐Adl, Nour E. A. Abd El‐Sattar

2020Bioorganic Chemistry91 citationsDOI

Topics & Concepts

ChemistrySorafenibIC50Cell cultureStereochemistryDocking (animal)DoxorubicinCancer cellPharmacologyIn vitroCancerBiochemistryCancer researchChemotherapyBiologyMedicineGeneticsHepatocellular carcinomaNursingSynthesis and biological activityEnzyme function and inhibitionBioactive Compounds and Antitumor Agents
Design, green synthesis, molecular docking and anticancer evaluations of diazepam bearing sulfonamide moieties as VEGFR-2 inhibitors | Litcius