Discovery of novel 2-substituted 2, 3-dihydroquinazolin-4(1H)-one derivatives as tubulin polymerization inhibitors for anticancer therapy: The in vitro and in vivo biological evaluation
Cai Shi, Boning Yang, Zhaolong He, Jingxiang Yang, Jingxiang Yang, Ling Li, Jian Song, Shiqiang Xu, Wei Song, Jian Yang, Jian Yang, Jian Yang, Jian Yang
Topics & Concepts
ChemistryIn vitroTubulinIn vivoApoptosisDocking (animal)MicrotubuleCell cycleCell cycle checkpointCell cultureStereochemistryPharmacologyBiochemistryCell biologyBiologyBiotechnologyNursingMedicineGeneticsQuinazolinone synthesis and applicationsSynthesis and biological activityCancer therapeutics and mechanisms