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Improving physicochemical properties of Ibrutinib with cocrystal strategy based on structures and natures of the carboxylic acid co-formers

Xiangjun Shi, Chao Wang, Qifeng Chen, Shuimei Shen, Shengjie Song, Xiyue Zhou

2021Journal of Drug Delivery Science and Technology22 citationsDOI

Topics & Concepts

CocrystalThermogravimetric analysisPowder diffractionSolubilityCrystallizationHydrogen bondDifferential scanning calorimetryDissolutionIbrutinibChemistryMaterials scienceCrystallographyOrganic chemistryMoleculeLeukemiaInternal medicineThermodynamicsMedicinePhysicsChronic lymphocytic leukemiaCrystallization and Solubility StudiesQuinazolinone synthesis and applicationsEnzyme Structure and Function
Improving physicochemical properties of Ibrutinib with cocrystal strategy based on structures and natures of the carboxylic acid co-formers | Litcius