Structural analysis of hERG channel blockers and the implications for drug design
Sara AlRawashdeh, Suryanarayanan Chandrasekaran, Khaled Barakat
Topics & Concepts
hERGCardiotoxicityPharmacologyDrugDrug discoveryPotassium channelChemistryLong QT syndromeComputational biologyMedicineBiologyBiochemistryBiophysicsToxicityQT intervalOrganic chemistryInternal medicineCardiac electrophysiology and arrhythmiasReceptor Mechanisms and SignalingComputational Drug Discovery Methods