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Discovery of anti-hepatoma agents from 1,4,5,6,7,8-hexahydropyrido[4,3-d]pyrimidine by inhibiting PI3K/AKT/NF-κB pathway activation

Yan-Qiu Zhou, Yue Sun, Hanlin Luo, Zhongfei Gao, Hongqin Zhang, Qingguo Meng, Xianyong Bai, Gui‐Ge Hou, Yun Hou

2021European Journal of Medicinal Chemistry23 citationsDOI

Topics & Concepts

ChemistryPI3K/AKT/mTOR pathwayProtein kinase BPhosphorylationPyrimidineApoptosisToxicityDocking (animal)Caspase 3NF-κBCancer researchCell biologyBiochemistryProgrammed cell deathBiologyNursingOrganic chemistryMedicineQuinazolinone synthesis and applicationsCytokine Signaling Pathways and InteractionsCancer Mechanisms and Therapy
Discovery of anti-hepatoma agents from 1,4,5,6,7,8-hexahydropyrido[4,3-d]pyrimidine by inhibiting PI3K/AKT/NF-κB pathway activation | Litcius