Targeting cyclin-dependent kinases: From pocket specificity to drug selectivity
Yaoguang Huang, Wenwu Liu, Changhao Zhao, Xiaoyu Shi, Qingchun Zhao, Jing‐Ming Jia, An‐Hua Wang, An‐Hua Wang
Topics & Concepts
Cyclin-dependent kinaseSelectivityKinaseChemistryDrug developmentCyclinDrugComputational biologyDrug discoveryBiochemistryPharmacologyBiologyGeneCell cycleCatalysisCancer-related Molecular PathwaysProtein Degradation and InhibitorsAdvanced Breast Cancer Therapies