Tyrosol 1,2,3-triazole analogues as new acetylcholinesterase (AChE) inhibitors
Guilherme Mateus Bousada, Bianca Lana de Sousa, Gabriela Milane Furlani, Ana Paula Agrizzi, Priscila Gonçalves Ferreira, João Paulo Viana Leite, Tiago Antônio de Oliveira Mendes, Eduardo Vinícius Vieira Varejão, Eduardo Jorge Pilau, Marcelo Henrique dos Santos
Topics & Concepts
AcetylcholinesteraseTyrosolChemistryAchéIC50Docking (animal)StereochemistryTacrineEnzymeTriazoleBiochemistryIn vitroOrganic chemistryMedicineAntioxidantNursingCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsSynthesis and biological activity