Discovery of novel artemisinin-sulfonamide hybrids as potential carbonic anhydrase IX inhibitors with improved antiproliferative activities
Ran An, Bin Lin, Shuang Zhao, Chun Cao, Yuanxin Wang, Xue Cheng, Yichuang Liu, Mengbi Guo, Hang Xu, Yitong Wang, Zhuang Hou, Chun Guo
Topics & Concepts
ChemistryCarbonic anhydraseArtemisininIC50CytotoxicityCarbonic Anhydrase ICell cultureExtracellularGrowth inhibitionHeLaDocking (animal)BiochemistryCytotoxic T cellCarbonic anhydrase IIIn vitroEnzymePlasmodium falciparumBiologyMedicineNursingGeneticsImmunologyMalariaEnzyme function and inhibitionSynthesis and Catalytic ReactionsCholinesterase and Neurodegenerative Diseases