Discovery of novel liver X receptor inverse agonists as lipogenesis inhibitors
Ziyang Chen, Hao Chen, Zizhen Zhang, Peng Ding, Xin Yan, Yanwen Li, Songxuan Zhang, Qiong Gu, Huihao Zhou, Jun Xu
Topics & Concepts
Liver X receptorChemistryInverse agonistLipogenesisAgonistAgonismNuclear receptorBiochemistryReceptorPharmacologyTranscription factorLipid metabolismBiologyGenePolitical sciencePoliticsLawCholesterol and Lipid MetabolismDrug Transport and Resistance MechanismsPeroxisome Proliferator-Activated Receptors