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Discovery, synthesis and biological evaluation of novel isoquinoline derivatives as potent indoleamine 2, 3-dioxygenase 1 and tryptophan 2, 3-dioxygenase dual inhibitors

Zhiqian Lin, Xiang-Li Ning, Ruizhi Lai, Li Hai, Ruifang Nie, Li Guo, Guo‐Bo Li, Zhongzhen Yang, Yong Wu

2024European Journal of Medicinal Chemistry11 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryIndoleamine 2,3-dioxygenaseIsoquinolineDioxygenaseTryptophanBiochemistryStereochemistryEnzymeAmino acidTryptophan and brain disordersPharmacological Receptor Mechanisms and EffectsCyclopropane Reaction Mechanisms
Discovery, synthesis and biological evaluation of novel isoquinoline derivatives as potent indoleamine 2, 3-dioxygenase 1 and tryptophan 2, 3-dioxygenase dual inhibitors | Litcius