Litcius/Paper detail

Development of a highly potent and selective degrader of LRRK2

John M. Hatcher, Monika Zwirek, Adil R. Sarhan, Prasanna S. Vatsan, Francesca Tonelli, Dario R. Alessi, Paul Davies, Nathanael S. Gray

2023Bioorganic & Medicinal Chemistry Letters17 citationsDOIOpen Access PDF

Topics & Concepts

LRRK2NeurodegenerationKinaseChemistryScaffold proteinDrug discoveryCell biologyPharmacologyBiochemistrySignal transductionMutationDiseaseBiologyGeneMedicineInternal medicineProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysSignaling Pathways in Disease
Development of a highly potent and selective degrader of LRRK2 | Litcius