Litcius/Paper detail

Dual Photochemical H‐Atom Transfer and Cobalt Catalysis for the Desaturative Synthesis of Phenols from Cyclohexanones

Henry P. Caldora, Zhenhua Zhang, Michael J. Tilby, Oliver Turner, Daniele Leonori

2023Angewandte Chemie International Edition39 citationsDOIOpen Access PDF

Abstract

Abstract Phenols are integral aromatic molecules widely encountered in the structure of natural products and routinely utilised for the synthesis of high‐value materials. Accessing highly substituted derivatives can often be difficult, especially when their functionalization pattern does not match the intrinsic reactivity leveraged by electrophilic aromatic substitution (S E Ar) chemistry. Here, we provide an alternative and mechanistically distinct approach for phenol synthesis using saturated cyclohexanone precursors. This process operates at ambient temperature, under simple purple light irradiation, and features a dual catalytic manifold carrying four sequential H‐atom transfer processes.

Topics & Concepts

CobaltCatalysisPhotochemistryPhenolsChemistryDual (grammatical number)Atom (system on chip)Organic chemistryComputer scienceArtLiteratureEmbedded systemRadical Photochemical ReactionsCatalytic C–H Functionalization MethodsAsymmetric Hydrogenation and Catalysis