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Allosteric modulation of ryanodine receptor RyR1 by nucleotide derivatives

Spencer CHOLAK, James W. Saville, Xing Zhu, Alison Berezuk, Katharine S. Tuttle, Omid Haji‐Ghassemi, Francisco Alvarado, Filip Van Petegem, Sriram Subramaniam

2023Structure27 citationsDOIOpen Access PDF

Topics & Concepts

RYR1Ryanodine receptorAllosteric regulationBiophysicsChemistryAdenosine triphosphateEndoplasmic reticulumBiochemistryAdenosineAdenine nucleotideNucleotideCell biologyReceptorBiologyGeneIon channel regulation and functionCardiac electrophysiology and arrhythmiasCalcium signaling and nucleotide metabolism
Allosteric modulation of ryanodine receptor RyR1 by nucleotide derivatives | Litcius