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Ibrutinib Blocks YAP1 Activation and Reverses BRAF Inhibitor Resistance in Melanoma Cells

Sean A. Misek, Patrick Newbury, Evgenii Chekalin, Shreya Paithankar, Andrea I. Doseff, Bin Chen, Kathleen A. Gallo, Richard R. Neubig

2021Molecular Pharmacology16 citationsDOIOpen Access PDF

Topics & Concepts

IbrutinibMelanomaCancer researchChemistryMedicinePharmacologyInternal medicineLeukemiaChronic lymphocytic leukemiaMelanoma and MAPK PathwaysHippo pathway signaling and YAP/TAZPI3K/AKT/mTOR signaling in cancer
Ibrutinib Blocks YAP1 Activation and Reverses BRAF Inhibitor Resistance in Melanoma Cells | Litcius