Refinement of safety and efficacy of anti-cancer chemotherapeutics by tailoring their site-specific intracellular bioavailability through transporter modulation
Pooja Dhakne, Megha Pillai, Sonam Mishra, Bappaditya Chatterjee, Rakesh Kumar Tekade, Pinaki Sengupta
Topics & Concepts
EffluxTransporterBioavailabilityPharmacologyATP-binding cassette transporterIntracellularDrug discoveryMultiple drug resistanceDrugSolute carrier familyBiologyDrug resistanceBioinformaticsBiochemistryGeneGeneticsDrug Transport and Resistance MechanismsPharmacological Effects and Toxicity StudiesAmino Acid Enzymes and Metabolism