Litcius/Paper detail

Development of Hydrogen Sulfide-Releasing Carbonic Anhydrases IX- and XII-Selective Inhibitors with Enhanced Antihyperalgesic Action in a Rat Model of Arthritis

Alessandro Bonardi, Laura Micheli, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Paola Gratteri, Alessio Nocentini, Claudiu T. Supuran

2022Journal of Medicinal Chemistry21 citationsDOIOpen Access PDF

Abstract

S donor, CAI fragment, or their co-administration.

Topics & Concepts

ChemistryArthritisIn vivoPharmacologyIn vitroHydrogen sulfidePotencyBiochemistryInternal medicineMedicineOrganic chemistryBiologyBiotechnologySulfurEnzyme function and inhibitionPhenothiazines and Benzothiazines Synthesis and ActivitiesMast cells and histamine