Synthesis, characterization and biological evaluation of novel azo fused 2,3-dihydro-1H-perimidine derivatives: In vitro antibacterial, antibiofilm, anti-quorum sensing, DFT, in silico ADME and Molecular docking studies
N. Nagasundaram, Chinnasamy Govindhan, Sivagiri Sumitha Sivagiri Sumitha, Nagarajan Sedhu, Krishnan Raguvaran, Santhosh Sigamani, Appaswami Lalitha
Topics & Concepts
ChemistryADMEQuorum sensingIn silicoSwarming motilityBiofilmChromobacterium violaceumAntibacterial activityCombinatorial chemistryPseudomonas aeruginosaDocking (animal)In vitroStereochemistryBiochemistryBacteriaGeneGeneticsBiologyVirulenceNursingMedicineSynthesis and Biological EvaluationPhenothiazines and Benzothiazines Synthesis and ActivitiesQuinazolinone synthesis and applications