Glutathione-responsive PROTAC for targeted degradation of ERα in breast cancer cells
Z. Zhou, Heli Fan, Dehao Yu, Fengying Shi, Qianqian Li, Zhenjian Zhang, Xiaolu Wang, Xuejun Zhang, Cheng Dong, Huabing Sun, Wenyi Mi
Topics & Concepts
GlutathioneChemistryEstrogen receptorCancer researchCancer cellBreast cancerCancerTumor microenvironmentProteolysisEstrogenPharmacologyBiochemistryInternal medicineMedicineEnzymeProtein Degradation and InhibitorsPeptidase Inhibition and AnalysisUbiquitin and proteasome pathways