Litcius/Paper detail

Interaction study with DNA/HSA, anti-topoisomerase IIα, cytotoxicity and in vitro antiproliferative evaluations and molecular docking of indole-thiosemicarbazone compounds

Íris Trindade Tenório Jacob, Iranildo José da Cruz Filho, Josival Emanuel Ferreira Alves, Felipe de Melo Souza, Rafael David Souto de Azevedo, Diego Santa Clara Marques, Túlio Ricardo Couto de Lima Souza, Keriolaine Lima dos Santos, Maíra Galdino da Rocha Pitta, Moacyr Jesus Barreto de Melo Rêgo, Jamerson Ferreira de Oliveira, Sinara Mônica Vitalino de Almeida, Maria do Carmo Alves de Lima

2023International Journal of Biological Macromolecules16 citationsDOI

Topics & Concepts

TopoisomeraseChemistryCytotoxicityDocking (animal)Indole testIC50StereochemistryIn vitroBinding constantHuman serum albuminSemicarbazoneJurkat cellsEnzymeBiochemistryMolecular modelBinding siteBiologyT cellImmunologyNursingMedicineImmune systemCancer therapeutics and mechanismsPharmacogenetics and Drug MetabolismSynthesis and biological activity