Synthesis and evaluation of the epithelial-to- mesenchymal inhibitory activity of indazole-derived imidazoles as dual ALK5/p38α MAP inhibitors
Yue Ying Liu, Zhen Guo, Jing Ying Wang, Huimin Wang, Jun Qi, Juan Ma, Hu‐Ri Piao, Cheng Hua Jin, Xuejun Jin
Topics & Concepts
ChemistryEpithelial–mesenchymal transitionp38 mitogen-activated protein kinasesKinaseVimentinProtein kinase ABlotTransforming growth factorMesenchymal stem cellMolecular biologyCell biologyBiochemistryImmunohistochemistryTransition (genetics)BiologyImmunologyGeneTGF-β signaling in diseasesBone Metabolism and DiseasesCytokine Signaling Pathways and Interactions