Litcius/Paper detail

Derivatization based on tetrazine scaffolds: synthesis of tetrazine derivatives and their biomedical applications

Hongbao Sun, Qinghe Xue, Chang Zhang, Haoxing Wu, Ping Feng

2021Organic Chemistry Frontiers39 citationsDOI

Abstract

The recent advances in tetrazine scaffold-based derivatizations have been summarized. The advantages and limitations of derivatization methods and applications of the developed tetrazine derivatives in bioorthogonal chemistry have been highlighted.

Topics & Concepts

TetrazineChemistryDerivatizationCombinatorial chemistryOrganic chemistryHigh-performance liquid chromatographyClick Chemistry and ApplicationsChemical Synthesis and AnalysisSynthesis and Biological Evaluation