Identification and optimization of a novel series of selective PIP5K inhibitors
David Andrews, Sharon Cartic, Sabina Cosulich, Nullin Divecha, Paul Faulder, Vikki Flemington, Oliver Kern, Jason G. Kettle, Ellen MacDonald, Jennifer C. McKelvie, Kurt G. Pike, Bryan Roberts, Rachel Rowlinson, James M. Smith, Martin L. Stockley, Martin E. Swarbrick, Iris Treinies, Michael J. Waring
Topics & Concepts
Drug discoveryComputational biologyChemistryIdentification (biology)Small moleculeKinaseBiochemistryBiologyBotanyCellular transport and secretionProtein Kinase Regulation and GTPase SignalingEndoplasmic Reticulum Stress and Disease