Litcius/Paper detail

PTG-0861: A novel HDAC6-selective inhibitor as a therapeutic strategy in acute myeloid leukaemia

Justyna M. Gawel, Andrew E. Shouksmith, Yasir S. Raouf, Nabanita Nawar, Krimo Toutah, Shazreh Bukhari, Pimyupa Manaswiyoungkul, Olasunkanmi O. Olaoye, Johan Israelian, Tudor B. Radu, Aaron D. Cabral, Diana Sina, Abootaleb Sedighi, Elvin D. de Araujo, Patrick T. Gunning

2020European Journal of Medicinal Chemistry41 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryHDAC6DruggabilityCancer researchPharmacologyHistone deacetylaseBiochemistryBiologyHistoneGeneHistone Deacetylase Inhibitors ResearchProtein Degradation and InhibitorsPeptidase Inhibition and Analysis