PTG-0861: A novel HDAC6-selective inhibitor as a therapeutic strategy in acute myeloid leukaemia
Justyna M. Gawel, Andrew E. Shouksmith, Yasir S. Raouf, Nabanita Nawar, Krimo Toutah, Shazreh Bukhari, Pimyupa Manaswiyoungkul, Olasunkanmi O. Olaoye, Johan Israelian, Tudor B. Radu, Aaron D. Cabral, Diana Sina, Abootaleb Sedighi, Elvin D. de Araujo, Patrick T. Gunning
Topics & Concepts
ChemistryHDAC6DruggabilityCancer researchPharmacologyHistone deacetylaseBiochemistryBiologyHistoneGeneHistone Deacetylase Inhibitors ResearchProtein Degradation and InhibitorsPeptidase Inhibition and Analysis