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Squaramide-catalyzed asymmetric Michael/cyclization of 4-isothiocyanato pyrazolones and α,β-unsaturated ketones

Wenjing Gong, Xin Du, Wenyao Wang, Wande Zhang, Baomin Wang

2021Tetrahedron Letters12 citationsDOI

Topics & Concepts

SquaramideStereocenterPyrazolonesChemistryMichael reactionPyrazoloneOrganocatalysisSubstrate (aquarium)Cascade reactionCatalysisEnantioselective synthesisScope (computer science)Combinatorial chemistryOrganic chemistryMedicinal chemistryOceanographyProgramming languageComputer scienceGeologyAsymmetric Synthesis and CatalysisChemical Synthesis and ReactionsSynthesis and Catalytic Reactions
Squaramide-catalyzed asymmetric Michael/cyclization of 4-isothiocyanato pyrazolones and α,β-unsaturated ketones | Litcius