Discovery of a Small Molecule Drug Candidate for Selective NKCC1 Inhibition in Brain Disorders
Annalisa Savardi, Marco Borgogno, Roberto Narducci, Giuseppina La Sala, José Antonio Ortega, Maria Summa, Andrea Armirotti, Rosalia Bertorelli, Andrea Contestabile, Marco De Vivo, Laura Cancedda
Topics & Concepts
BumetanidePharmacologyDrugDiureticTransporterDrug discoveryPharmacogenomicsMedicineIntracellularDrug candidateToxicityHomeostasisBioinformaticsChemistryBiologyInternal medicineGeneBiochemistryMembraneIon transporterGenetics and Neurodevelopmental DisordersIon Transport and Channel RegulationEpilepsy research and treatment