Discovery of a highly potent CECR2 bromodomain inhibitor with 7H-pyrrolo[2,3-d] pyrimidine scaffold
Haibo Lu, Tian Lu, Shijia Zu, Z. H. Duan, Yiman Guang, Qi Li, Jingyi Ma, Dongying Chen, Bo Li, Wenchao Lu, Hualiang Jiang, Cheng Luo, Deyong Ye, Kaixian Chen, Hua Lin
Topics & Concepts
BromodomainChemistryPyrimidineChromatinDocking (animal)Chromatin remodelingComputational biologyStereochemistryBiochemistryEpigeneticsGeneBiologyMedicineNursingProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsUbiquitin and proteasome pathways