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Activation of Phospholipase C β by Gβγ and Gαq Involves C-Terminal Rearrangement to Release Autoinhibition

Isaac J. Fisher, Meredith L. Jenkins, Gregory G. Tall, John E. Burke, Alan V. Smrcka

2020Structure42 citationsDOIOpen Access PDF

Topics & Concepts

Gq alpha subunitCTDPhospholipase CChemistryG protein-coupled receptorC-terminusDiacylglycerol kinasePhospholipaseG proteinBiophysicsStereochemistryBiochemistryEnzymeReceptorBiologyProtein kinase CAmino acidGeologyOceanographyProtein Kinase Regulation and GTPase SignalingReceptor Mechanisms and SignalingMetabolism, Diabetes, and Cancer
Activation of Phospholipase C β by Gβγ and Gαq Involves C-Terminal Rearrangement to Release Autoinhibition | Litcius