Design, synthesis and anti-diabetic activity of novel 1, 2, 3-triazole-5-carboximidamide derivatives as dipeptidyl peptidase-4 inhibitors
Hossein Fasihi Dastjerdi, Nima Naderi, Manijeh Nematpour, Elham Rezaee, Mohammad Mahboubi‐Rabbani, Melika Ebrahimi, Samaneh Hosseinipoor, Omid Hosseini, Sayyed Abbas Tabatabai
Topics & Concepts
ChemistrySitagliptinDipeptidyl peptidaseIC50Dipeptidyl peptidase-4EnzymePharmacologyDiabetes mellitusInhibitory postsynaptic potentialGlucagonTriazolePancreasType 2 Diabetes MellitusEndocrinologyBiochemistryType 2 diabetesIn vitroHormoneOrganic chemistryMedicinePeptidase Inhibition and AnalysisDiabetes Treatment and ManagementAdenosine and Purinergic Signaling