Design and synthesis of quinoxaline-1,3,4-oxadiazole hybrid derivatives as potent inhibitors of the anti-apoptotic Bcl-2 protein
Yukari Ono, Masayuki Ninomiya, Daiki Kaneko, Amol D. Sonawane, Taro Udagawa, Kaori Tanaka, Atsuyoshi Nishina, Mamoru Koketsu
Topics & Concepts
QuinoxalineChemistryOxadiazoleCytotoxicityApoptosisMorpholinePiperidineCell culturePiperazineCell growthBiochemistryStereochemistryIn vitroBiologyMedicinal chemistryOrganic chemistryGeneticsSynthesis and Biological EvaluationCAR-T cell therapy researchCancer therapeutics and mechanisms