Litcius/Paper detail

Unique Pharmacological Properties of the Kappa Opioid Receptor Signaling Through Gαz as Shown with Bioluminescence Resonance Energy Transfer

Miriam Barnett, Brian I. Knapp, Jean M. Bidlack

2020Molecular Pharmacology13 citationsDOIOpen Access PDF

Topics & Concepts

G proteinκ-opioid receptorHeterotrimeric G proteinChemistryDynorphinReceptorμ-opioid receptorOpioidIntrinsic activityDynorphin AG protein-coupled receptorPharmacologyAgonistStereochemistryBiochemistryOpioid peptideBiologyReceptor Mechanisms and SignalingNeuropeptides and Animal PhysiologyPharmacological Receptor Mechanisms and Effects