Molecular basis for anti-insomnia drug design from structure of lemborexant-bound orexin 2 receptor
Hidetsugu Asada, Dohyun Im, Yunhon Hotta, Satoshi Yasuda, Takeshi Murata, Ryoji Suno, So Iwata
Topics & Concepts
ReceptorOrexinPharmacophoreOrexin receptorChemistryWakefulnessPharmacologyBiophysicsBiologyBiochemistryNeuroscienceNeuropeptideElectroencephalographySleep and Wakefulness ResearchCircadian rhythm and melatoninSleep and related disorders