Binding sites and design strategies for small molecule GLP-1R agonists
Haibo Zhang, Tianxiao Wu, Yong Wu, Yuran Peng, Xian Wei, Tao Lü, Yu Jiao
Topics & Concepts
Allosteric regulationSmall moleculeIncretinGlucagon-like peptide-1ChemistryReceptorPharmacologyComputational biologyDiabetes mellitusMedicineType 2 diabetesBiochemistryEndocrinologyBiologyReceptor Mechanisms and SignalingDiabetes Treatment and ManagementNeuropeptides and Animal Physiology