Molecular hybrids integrated with imidazole and hydrazone structural motifs: Design, synthesis, biological evaluation, and molecular docking studies
Michael Tapera, Hüseyin Kekeçmuhammed, Emin Sarıpınar, Murat Doğan, Burak Tüzün, Ümit M. Koçyiğit, Feyza Nur Çetin
Topics & Concepts
Protein Data Bank (RCSB PDB)ADMEChemistryImidazoleDocking (animal)Active siteHydrazoneIn silicoStereochemistryCarbonic anhydraseEnzymeBiochemistryIn vitroNursingGeneMedicineEnzyme function and inhibitionSynthesis and biological activityCholinesterase and Neurodegenerative Diseases