Rezatapopt (PC14586): A First-in-Class Small Molecule p53 Y220C Mutant Protein Stabilizer in Clinical Trials
Zonghui Ma, Qiang Shen, Jia Zhou
Topics & Concepts
ChemistryStabilizer (aeronautics)MutantSmall moleculeMoleculeBiochemistryStereochemistryGeneOrganic chemistryEngineeringMechanical engineeringCancer-related Molecular PathwaysUbiquitin and proteasome pathwaysMicrotubule and mitosis dynamics