Hypoxia-activated pro-drugs of the KDAC inhibitor vorinostat (SAHA)
Ewen D. D. Calder, Anna Skwarska, Deborah Sneddon, Lisa K. Folkes, Ishna N. Mistry, Stuart J. Conway, Ester M. Hammond
Topics & Concepts
ChemistryVorinostatHypoxia (environmental)MoietyHistone deacetylase inhibitorPharmacologyOxygenHydroxamic acidHistone deacetylaseCombinatorial chemistryStereochemistryBiochemistryHistoneOrganic chemistryMedicineGeneHistone Deacetylase Inhibitors ResearchProtein Degradation and InhibitorsAdenosine and Purinergic Signaling