Litcius/Paper detail

Inverse Drug Discovery identifies weak electrophiles affording protein conjugates

Gabriel M. Kline, Karina Nugroho, Jeffery W. Kelly

2022Current Opinion in Chemical Biology21 citationsDOIOpen Access PDF

Topics & Concepts

ElectrophileDrug discoveryDruggabilityChemistryCombinatorial chemistryContext (archaeology)Covalent bondProteomeComputational biologyChemical biologyBiochemistryBiologyOrganic chemistryGeneCatalysisPaleontologyClick Chemistry and ApplicationsChemical Synthesis and AnalysisProtein Degradation and Inhibitors