Discovery of natural catechol derivatives as covalent SARS-CoV-2 3CLpro inhibitors
Feng Wang, Donglan Liu, Dingding Gao, Jinwei Yuan, Jingxian Zhao, Jingxian Zhao, Shuai Yuan, Yixin Cen, Guo‐Qiang Lin, Jincun Zhao, Jincun Zhao, Ping Tian
Topics & Concepts
ChemistryCatecholBiochemistryCathepsin LIC50Natural productEnzymeProteasesPharmacologyBiologyIn vitroComputational Drug Discovery MethodsSynthesis and bioactivity of alkaloidsBiological Stains and Phytochemicals