Litcius/Paper detail

Discovery of novel and selective GPR17 antagonists as pharmacological tools for developing new therapeutic strategies in diabetes and obesity

Hu Zhu, Jason M. Conley, Karavadhi Surendra, Justin LaVigne, Val J. Watts, Hongmao Sun, Min Shen, Matthew D. Hall, Hongxia Ren, Samarjit Patnaik

2025European Journal of Medicinal Chemistry10 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryDrug discoveryDiabetes mellitusPharmacologyObesityInternal medicineEndocrinologyMedicineBiochemistryDiabetes Treatment and ManagementReceptor Mechanisms and SignalingPancreatic function and diabetes