Novel compounds with dual S1P receptor agonist and histamine H3 receptor antagonist activities act protective in a mouse model of multiple sclerosis
Faik Imeri, Bisera Stepanovska Tanturovska, Aleksandra Živković, Gaby Enzmann, Stephanie Schwalm, Josef Pfeilschifter, Thomas Homann, Burkhard Kleuser, Britta Engelhardt, Holger Stark, Andrea Huwiler
Topics & Concepts
Histamine H3 receptorAgonistPharmacologyAntagonistHistamineReceptor antagonistCompetitive antagonistReceptorChemistryInverse agonistMedicineBiochemistrySphingolipid Metabolism and SignalingMast cells and histamineCircadian rhythm and melatonin