Litcius/Paper detail

Design, synthesis and antitumor evaluations of nucleoside base hydroxamic acid derivatives as DNMT and HDAC dual inhibitors

Qinsheng Sun, Qiuzi Dai, Cunlong Zhang, Yan Chen, Lei Zhao, Zigao Yuan, Yuyang Jiang

2021Chinese Chemical Letters13 citationsDOI

Topics & Concepts

ChemistryHydroxamic acidHDAC1Histone deacetylaseDNA methyltransferaseAcetylationEpigeneticsMethyltransferaseNucleosideHistoneBiochemistryMethylationDNAStereochemistryGeneHistone Deacetylase Inhibitors ResearchEpigenetics and DNA MethylationAdenosine and Purinergic Signaling